Publications
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Publications
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2024
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Journal Article
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Structure-Based Design of CBP/EP300 Degraders: When Cooperativity Overcomes Affinity. JACS Au, 4(9):3466-3474.
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Gold(III) Auracycles Featuring C(sp$^3$)‐Au‐C(sp$^2$) Bonds: Synthesis and Mechanistic Insights into the Cycloauration Step. Angewandte Chemie Internationale Edition, 63(36):e202402798.
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(P^N^C) Ligands to Stabilize Gold(III): A Straightforward Access to Hydroxo, Formate, and Hydride Complexes. Inorganic Chemistry, 63(18):8390-8396.
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Nickel-catalysed enantioselective alkene dicarbofunctionalization enabled by photochemical aliphatic C–H bond activation. Nature Catalysis, 7(6):655-665.
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Asymmetric, Remote C(sp$^3$)−H Arylation via Sulfinyl‐Smiles Rearrangement. Angewandte Chemie Internationale Edition, 63(17):e202319158.
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Chiral arylsulfinylamides as reagents for visible light-mediated asymmetric alkene aminoarylations. Nature Chemistry, 16(4):607-614.
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Dual Nickel/Photoredox‐Catalyzed Asymmetric Carbamoylation of Benzylic C(sp$_3$)−H Bonds. Angewandte Chemie Internationale Edition, 63(12):e202313717.
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Discovery and Characterization of Active CBP/EP300 Degraders Targeting the HAT Domain. ACS Medicinal Chemistry Letters, 15(3):355-361.
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2023
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Journal Article
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Reevaluation of bromodomain ligands targeting BAZ2A. Protein Science, 32(9):e4752.
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Dual Nickel/Photoredox-Catalyzed Asymmetric Carbosulfonylation of Alkenes. Journal of the American Chemical Society, 145(23):12532-12540.
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Nickel-Catalyzed Enantioselective Electrochemical Reductive Cross-Coupling of Aryl Aziridines with Alkenyl Bromides. Journal of the American Chemical Society, 145(11):6270-6279.
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2022
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Journal Article
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Synthesis of Cyclometalated Gold(III) Complexes via Catalytic Rhodium to Gold(III) Transmetalation. Angewandte Chemie Internationale Edition, 61(20):e202116755.
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2021
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Journal Article
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Diaryl Ether Formation Merging Photoredox and Nickel Catalysis. Organometallics, 40(14):2188-2193.
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Asymmetric, visible light-mediated radical sulfinyl-Smiles rearrangement to access all-carbon quaternary stereocentres. Nature Chemistry, 13(4):327-334.
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Synthesis and Characterization of Bidentate (P^N)Gold(III) Fluoride Complexes: Reactivity Platforms for Reductive Elimination Studies. Angewandte Chemie Internationale Edition, 60(8):4164-4168.
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Nickel‐Catalyzed Asymmetric Synthesis of α‐Arylbenzamides. Angewandte Chemie Internationale Edition, 60(3):1605-1609.
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Chelation-assisted C–C bond activation of biphenylene by gold(i) halides. Chemical Science, 12(45):15084-15089.
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2020
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Journal Article
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Phosphorescent K$^3$ -(N^C^C)-Gold(III) Complexes: Synthesis, Photophysics, Computational Studies and Application to Solution-Processable OLEDs. Chemistry - A European Journal, 26(72):17604-17612.
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[C^N]‐Alkenyl Gold(III) Complexes by Proximal Ring‐Opening of (2‐Pyridyl)alkylidenecyclopropanes: Mechanistic Insights. Angewandte Chemie Internationale Edition, 59(45):20049-20054.
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Mechanistic Insights into C(sp2)−C(sp)N Reductive Elimination from Gold(III) Cyanide Complexes. Angewandte Chemie Internationale Edition, 59(41):17881-17886.
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Hitting a Moving Target: Simulation and Crystallography Study of ATAD2 Bromodomain Blockers. ACS Medicinal Chemistry Letters, 11(8):1573-1580.
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Asymmetric Ni-Catalyzed Radical Relayed Reductive Coupling. Journal of the American Chemical Society, 142(31):13515-13522.
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Highly Efficient Green Solution Processable Organic Light-Emitting Diodes Based on a Phosphorescent K$^3$-(N^C^C)Gold(III)-Alkynyl Complex. Chemistry of Materials, 32(4):1605-1611.
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Understanding the mechanism of action of pyrrolo[3,2-b]quinoxaline-derivatives as kinase inhibitors. RSC Medicinal Chemistry, 11(6):665-675.
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2019
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Journal Article
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Ni-Catalyzed Reductive Dicarbofunctionalization of Nonactivated Alkenes: Scope and Mechanistic Insights. Journal of the American Chemical Society, 141(35):13812-13821.
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Dual Photoredox/Nickel‐Catalyzed Three‐Component Carbofunctionalization of Alkenes. Angewandte Chemie Internationale Edition, 58(35):12286-12290.
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K$^3$‐(N^C^C)Gold(III) Carboxylates: Evidence for Decarbonylation Processes. Angewandte Chemie Internationale Edition, 131(27):9162-9165.
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Oxidant speciation and anionic ligand effects in the gold-catalyzed oxidative coupling of arenes and alkynes. Chemical Science, 10(36):8411-8420.
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2018
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Journal Article
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Binding Motifs in the CBP Bromodomain: An Analysis of 20 Crystal Structures of Complexes with Small Molecules. ACS Medicinal Chemistry Letters, 9(9):929-934.
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Structural Analysis of Small-Molecule Binding to the BAZ2A and BAZ2B Bromodomains. ChemMedChem, 13(14):1479-1487.
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Visible Light Mediated, Redox Neutral Remote 1,6-Difunctionalizations of Alkenes. ACS Catalysis, 8(7):6401-6406.
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Transforming Olefins into Dinucleophiles. CHIMIA International Journal for Chemistry, 72(4):212-215.
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Iriomoteolides: novel chemical tools to study actin dynamics. Chemical Science, 9(15):3793-3802.
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Gold-catalyzed oxidative aminoesterification of unactivated alkenes. Monatshefte für Chemie / Chemical Monthly, 149(4):749-754.
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Chemical Space Expansion of Bromodomain Ligands Guided by in Silico Virtual Couplings (AutoCouple). ACS Central Science, 4(2):180-188.
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2017
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Journal Article
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Cyclometalated gold(III) complexes: synthesis, reactivity, and physicochemical properties. Angewandte Chemie Internationale Edition, 56(8):1994-2015.
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Expeditious diastereoselective synthesis of elaborated ketones via remote Csp3–H functionalization. Nature Communications, 8:13832.
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Visible-light-mediated remote aliphatic C−H functionalizations through a 1,5-hydrogen transfer cascade. Angewandte Chemie Internationale Edition, 56(7):1881-1884.
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Stereoselective carboperfluoroalkylation of internal alkynes: mechanistic insights. Topics in Catalysis, 60(8):545-553.
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Nickel-catalyzed reductive dicarbofunctionalization of alkenes. Journal of the American Chemical Society, 139(20):6835-6838.
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Nickel-catalyzed intermolecular carbosulfonylation of alkynes via sulfonyl radicals. Angewandte Chemie Internationale Edition, 56(33):9949-9952.
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γ-functionalizations of amines through visible-light-mediated, redox-neutral C−C bond cleavage. Angewandte Chemie Internationale Edition, 56(35):10521-10524.
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The first gold(III) formate: evidence for β-hydride elimination. Angewandte Chemie Internationale Edition, 56(42):12862-12865.
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A gold- and brønsted acid catalytic interplay towards the synthesis of highly substituted tetrahydrocarbazoles. Helvetica Chimica Acta, 100(3):e1600333.
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2016
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Journal Article
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Gold-catalyzed direct oxidative arylation with boron coupling partners. Angewandte Chemie Internationale Edition, 56(4):1021-1025.
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Evidence for direct transmetalation of AuIII–F with boronic acids. Journal of the American Chemical Society, 138(42):13790-13793.
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In vivo performance and properties of tamoxifen metabolites for CreERT2 control. PLoS ONE, 11(4):e0152989.
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The “Gatekeeper” residue influences the mode of binding of acetyl indoles to bromodomains. Journal of Medicinal Chemistry, 59(7):3087-3097.
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Palladium-catalyzed incorporation of atmospheric CO2: efficient synthesis of functionalized oxazolidinones. Chemical Science, 7(6):3914-3918.
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Au–Pd bimetallic catalysis: the importance of anionic ligands in catalyst speciation. Journal of the American Chemical Society, 138(10):3266-3269.
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